Gịnị bụArtesunates?
Artesunate bụ ọgwụ mgbochi ịba. Ọ bụ hemisuccinate na-agbaze mmiri nke dihydroartemisinin.
Artemisinin bụ sesquiterpene lactone dịpụrụ adịpụ na Artemisia annua, ogwu nke ejirila na China mee ihe maka ọgwụgwọ ịba.
Artesunates na metabolite dihydroartemisinin ya na-arụ ọrụ bụ schizonticide ọbara dị ike, na-arụ ọrụ megide mgbanaka mgbanaka nke nje. Artesunate dị mma maka ọgwụgwọ ọrịa ịba siri ike, gụnyere ịba ụbụrụ. Ọ na-arụkwa ọrụ megide chloroquine na mefloquine na-eguzogide ụdị P. falciparum. Ọ naghị akwụsi ike na ngwọta na-anọpụ iche, ya mere ọ dị naanị maka injections dị ka artesunic acid. A ghaghị ịkwado usoro injectable ozugbo tupu ejiri ya na 5% (w / v) sodium bicarbonate ngwọta iji mepụta nnu sodium artesunate.
Aha | Artesunates |
CAS NO. | 88495-63-0 |
Usoro ihe omimi | C19H28O8 |
Nyocha | 99% |
Njirimara | White crystalline ntụ ntụ |
Ibu molekụla | 384.42 |
1.Artesunate nwere ọrụ ịchịkwa ịba vivax na mgbaàmà ịba falciparum, yana ọgwụgwọ ahụhụ na-eguzogide chloroquine.
2. Artesunate nwere ọrụ nke oxidant. A na-ebelata artemisinin site na catalase, dithiothreitol na alfa tocopherol.
3.Artesunate nwere ọrụ nke antibacterial, artemisinin nwere mmetụta nje virus na-egbochi nje.
4.Artesunate na ọrụ nke mgbochi parasaiti, artemisinin na ọrụ nke mgbochi schistosomiasis na leptospirosis.
Nyocha | Nkọwapụta | Nsonaazụ |
Ọdịdị | Gbanyụọ ntụ ntụ ọcha | Na-akwado |
Isi | Njirimara | Na-akwado |
nkọwapụta | Nobilatin 98% | Na-akwado |
Sieve analysis | 100% gafere 80 mesh | Na-akwado |
Ọnwụ na ihicha | ≤5.0% | Na-akwado |
Ihe fọdụrụ na mgbanye | ≤5.0% | Na-akwado |
Ọla dị arọ | Na-akwado | |
Dị ka | ≤1pm | Na-akwado |
Ihe mgbaze fọdụrụnụ | EP2000 | Na-akwado |
Mgbochi ahịhịa | Ihe ọjọọ | Na-akwado |
Microbiology | ||
Ngụkọta ọnụ ọgụgụ efere | Na-akwado | |
Yist & ebu | Na-akwado | |
E.Coli | Ihe ọjọọ | Na-akwado |
Salmonella | Ihe ọjọọ | Na-akwado |
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